Hui-fei Wang, Run Gan, Jing Zhou, Qi Liao, Tian-bao Wang, Cai-ling Zhong, Yuan-yuan Xiang, Hong-bo Lin, Xiang-nan Hu
2-(3-hydroxy-1-adamantyl)-2-oxoacetic acid (IV), a key intermediate of saxagliptin for type 2 diabetes mellitus (T2DM)
Diabetes
key intermediate
saxagliptin
optimization
one-pot method.